Isonicotinic acid explained

Isonicotinic acid or pyridine-4-carboxylic acid is an organic compound with the formula C5H4N(CO2H). It is a derivative of pyridine with a carboxylic acid substituent at the 4-position. It is an isomer of picolinic acid and nicotinic acid, which have the carboxyl group at the 2- and 3-position respectively compared to the 4-position for isonicotinic acid.

Production

On a commercial scale, isonicotinic acid, like other pyridine carboxylic acid is produced by ammoxidation of 4-picoline (4-methylpyridine) followed by hydrolysis of the resulting nitrile:

It is also produced by oxidation of 4-picoline with nitric acid.

Derivatives

Isonicotinic acids is a term loosely used for derivatives of isonicotinic acid. Hydrazide derivatives include isoniazid, iproniazid, and nialamide. Amide and ester derivatives include ethionamide and dexamethasone isonicotinate.

Its conjugate base forms coordination polymers[1] and MOFs[2] by binding metal ions through both the N and carboxylate.

See also

Notes and References

  1. 10.1016/j.ccr.2005.07.008 . Self-assembly directed by dinuclear zinc(II) macrocyclic species . 2006 . Huang . Wei . Zhu . Hai-Bin . Gou . Shao-Hua . Coordination Chemistry Reviews . 250 . 3–4 . 414–423 .
  2. 10.1021/jacs.8b07563 . Boosting Ethane/Ethylene Separation within Isoreticular Ultramicroporous Metal–Organic Frameworks . 2018 . Lin . Rui-Biao . Wu . Hui . Li . Libo . Tang . Xiao-Liang . Li . Zhiqiang . Gao . Junkuo . Cui . Hui . Zhou . Wei . Chen . Banglin . Journal of the American Chemical Society . 140 . 40 . 12940–12946 . 30216725 .