Salvianolic acids explained

Salvianolic acids are a group of polyphenolic acids consisting on several combinations of caffeic acid and danshensu (salvianic acid) through ester and enol bonds. Salvianolic acids are water-soluble components produced by many species of the genus Salvia, mainly extracted from Salvia miltiorrhiza.

Structural properties

More than 10 distinct salvianolic acids (Sal), identified by letters from A to J, have been recognized. Notably, Sal-A and Sal-B are the most abundant forms. The combination of danshensu and a caffeic acid derivative or caffeic acid dimer produces several kinds of skeletons. Sal-A is formed by a molecule of danshensu and a dimer of caffeic acid. Sal-B, on the other hand, is constituted by three molecules of danshensu and one molecule of caffeic acid. Sal-C results from the combination of two molecules of danshensu, while Sal-D is characterized as a dimer of caffeic acid.[1]

Biosynthesis and natural occurrence

The formation of salvianolic acids is closely linked to that of rosmarinic acid. They are primarily synthesized through the phenylpropanoid and tyrosine-derived branches of the phenolic acid biosynthetic pathway. Rosmarinic acid undergoes a not well-understood oxidative reaction to convert into Salvianolic acid B.[2] This reaction involves laccases, which are widely spread in many genera such as Arabidopsis, poplars, sorghum, etc., but appears to be highly expressed in Salvia miltiorrhiza and Salvia bowleyana.[3]

Notes and References

  1. Ma . Lunkun . Tang . Liling . Yi . Qian . 2019 . Salvianolic Acids: Potential Source of Natural Drugs for the Treatment of Fibrosis Disease and Cancer . Frontiers in Pharmacology . 10 . 97 . 10.3389/fphar.2019.00097 . free . 30842735 . 6391314 . 1663-9812.
  2. Zhou . Zheng . Li . Qing . Xiao . Liang . Wang . Yun . Feng . Jingxian . Bu . Qitao . Xiao . Ying . Hao . Kai . Guo . Meili . Chen . Wansheng . Zhang . Lei . 2021-03-18 . Multiplexed CRISPR/Cas9-Mediated Knockout of Laccase Genes in Salvia miltiorrhiza Revealed Their Roles in Growth, Development, and Metabolism . Frontiers in Plant Science . 12 . 647768 . 10.3389/fpls.2021.647768 . free . 1664-462X . 8014014 . 33815454.
  3. Li . Qing . Feng . Jingxian . Chen . Liang . Xu . Zhichao . Zhu . Yingjie . Wang . Yun . Xiao . Ying . Chen . Junfeng . Zhou . Yangyun . Tan . Hexin . Zhang . Lei . Chen . Wansheng . 2019 . Genome-Wide Identification and Characterization of Salvia miltiorrhiza Laccases Reveal Potential Targets for Salvianolic Acid B Biosynthesis . Frontiers in Plant Science . 10 . 435 . 10.3389/fpls.2019.00435 . free . 31024599 . 6463009 . 1664-462X.